Quantification of levetiracetam in plasma of neonates by ultra performance liquid chromatography-tandem mass spectrometry

Blonk, MI; van der Nagel, BC; Smit, LS; Mathot, RA

HERO ID

1037569

Reference Type

Journal Article

Year

2010

Language

English

PMID

20138814

HERO ID 1037569
In Press No
Year 2010
Title Quantification of levetiracetam in plasma of neonates by ultra performance liquid chromatography-tandem mass spectrometry
Authors Blonk, MI; van der Nagel, BC; Smit, LS; Mathot, RA
Journal Journal of Chromatography B: Analytical Technologies in the Biomedical and Life Sciences
Volume 878
Issue 7-8
Page Numbers 675-681
Abstract A sensitive and specific method using ultra performance liquid chromatography-tandem mass spectrometry (UPLC-MS/MS) was developed for the determination of levetiracetam (LEV) in plasma of neonates. A plasma aliquot of 50 microl was deproteinized by addition of 500 microl methanol which contained 5 microg/ml UCB 17025 as an internal standard. After centrifugation, 50 microl of supernatant was diluted with 1000 microl of 0.1% formic acid-10 mM ammonium formate in water (pH 3.5) (mobile phase solution A) and 2 microl was injected onto the UPLC-system. Compounds were separated on a Acquity UPLC BEH C(18) 2.1 mm x 100 mm column using gradient elution with mobile phase solution A and 0.1% formic acid in methanol (mobile phase solution B) with a flow rate of 0.4 ml/min and a total runtime of 4.0 min. LEV and the internal standard were detected using positive ion electrospray ionization followed by tandem mass spectrometry (ESI-MS/MS). The assay allowed quantification of LEV plasma concentrations in the range from 0.5 microg/ml to 150 microg/ml. Inter-assay inaccuracy was within +/-2.7% and inter-assay precision was less than 4.5%. Matrix effects were minor: the recovery of LEV was between 97.7% and 100%. The developed method required minimal sample preparation and less plasma sample volume compared to earlier published LC-MS/MS methods. The method was successfully applied in a clinical pharmacokinetic study in which neonates received intravenous administrations of LEV for the treatment of neonatal seizures.
Doi 10.1016/j.jchromb.2010.01.037
Pmid 20138814
Wosid WOS:000275565200008
Is Certified Translation No
Dupe Override No
Comments Source: Web of Science 000275565200008
Is Public Yes
Language Text English
Keyword Ultra performance liquid chromatography; Mass spectrometry; Levetiracetam; Plasma; Neonates; Pharmacokinetics
Is Qa No